Custom Peptides
Cayman Chemical N-BenzylpalmItamIde 10mg
A long-chain fatty acid amide isolated from the maca plant that moderately inhibits FAAH activity (44% inhibition at 500 µM); many members of this family demonstrate selective antiproliferative activity against diverse cancer cell lines
Cayman Chemical NdodecnoylLHomoserIn lac 10mg
A fluorescently tagged probe which allows the HSL molecule to be detected using fluorescence-based techniques
Cayman Chemical 2ImIno4methylpIperIdIna 10mg
2-Imino-4-methylpiperidine is a potent, general NOS inhibitor. It exhibits IC50 values of 0.1, 1.1, and 0.2 µM for inhibition of human iNOS, eNOS, and nNOS, respectively, at an arginine concentration of 30 µM.{5579}
Cayman Chemical HexnolamIno PAF C-16 10mg
Hexanolamino PAF C-16 is a PAF analog with mixed PAF receptor agonist/antagonist properties. In human monocyte-derived macrophages, it is an antagonist which inhibits the production of reactive oxygen species in response to PAF C-16.{367} On the other hand, in rabbit platelets and guinea pig macrophages, hexanolamino PAF C-16 is a partial agonist, and in guinea pig platelets it is a full agonist.{3786}
Cayman Chemical R-Docosahexaenyl-1-Hyd 10mg
A homolog of DHEA, characterized by the addition of an (R)-α-methyl group at the methylene carbon adjacent to the amide nitrogen
Cayman Chemical HydroxystIlbamIdInmethns 10mg
A fluorescent neuronal retrograde tracer and nucleic acid dye; labels the neuronal cell body as well as proximal dendrites; ex/em = 323/620 nm, respectively, when visualized in tissue sections; can be used to label DNA and RNA in fixed or unfixed dead cells; ex/em = 360/450 and 600 nm, respectively, when bound to DNA; ex/em = 360/450 nm, respectively, when bound to RNA
Cayman Chemical Rabeprazole sulfon 10mg
A metabolite of rabeprazole; has been found as an impurity in bulk preparations of rabeprazole
Cayman Chemical MELK-8ahydrochlorIde 10mg
A MELK inhibitor (IC50 = 0.002 µM); selective for MELK over FLT3, haspin, KIT, and PDGFRα, (IC50s = 0.18, 0.19, >10, and 0.42 µM, respectively), as well as a panel of 456 kinases at 1 µM; inhibits the proliferation of MDA-MB-468 and MCF-7 cells (IC50s = 0.11 and 3.68 µM)
Cayman Chemical PRfluoropentnsulfonIc ACD 10mg
A perfluoroalkyl substance; has been found as a contaminant in wastewater and breastmilk
Cayman Chemical KSL128114trIfluoroacetAT 10mg
A peptide syntenin inhibitor (Ki = 300 nM); reduces the percent viability of A2058 melanoma and patient-derived GBM cells in a concentration-dependent manner; increases animal survival time in a PDX mouse model of GBM using patient-derived GBM cells co-cultured with KSL-128114 prior to intracranial implantation at 50 µM
Cayman Chemical BIotInH10trIfluoroacetAT 10mg
A biotinylated form of H10; has been used in ELISA and co-immunoprecipitation assays to assess AGR2 levels in cancer cells
Cayman Chemical McaAVLQSGFRK DnpKNH2tr 10mg
A fluorogenic substrate for SARS-CoV Mpro; Mca is released upon cleavage by SARS-CoV Mpro and its fluorescence can be used to quantify SARS-CoV Mpro activity; ex/em = 328/420 nm, respectively
Cayman Chemical RPalmItoyl 1methyl Ethno 10mg
A synthetic analog of PEA which incorporates an (R)-methyl group vicinal to the alcohol on the ethanolamine moiety, which may protect the molecule from enzymatic hydrolysis, leading to prolonged duration of action and enhanced potency in vivo; expected to show enhancement of the inhibitory activity of PEA on mast cells and other cells known to express the CB2 receptor
Cayman Chemical MescalIn NBOMehydrochLRId 10mg
A derivative of mescaline having an N-(2-methoxybenzyl) addition at the amine
Cayman Chemical 4-EAPBhydrochlorIde 10mg
An analytical reference standard categorized as a benzofuran; intended for research and forensic applications